Cholinergic drugs
Anticholinergic drugs
Adrenergic drugs
Antiadrenergic drugs
Ganglion stimulant and blockers
Showing posts with label Autonomic Nervous System. Show all posts
Showing posts with label Autonomic Nervous System. Show all posts
Sunday, November 27, 2016
Ganglion stimulant and blockers classification
1)
Ganglionic Stimulants
a) Non-selective/muscarinic
agonists
Acetylcholine
Carbachol
Pilocarpine
Anticholinesterases
b)
Selective nicotinic agonists
Nicotine (low dose)
Lobeline
Dimethyl phenyl piperazinium iodide (DMPP)
Tetramethyl ammonium (TMA)
2)
Ganglion Blocking Agents
a)
Persistent depolarizing blockers
Nicotine (high dose)
Anticholinesterases (high dose)
b)
Competitive blockers
Trimethaphan
Mecamylamine
Hexamethonium
Pempidine
Pentolinium
Anti-adrenergic drugs classification
1) α Blockers
a) Non-equilibrium
type
Phenoxybenzamine
b)
Equilibrium type
i)
Non-selective
Ergot
alkaloids and derivatives
Ergotamine
Ergotoxine
Dihydroergotamine (DHE)
Dihydroergotoxine
Imidazolines
Phentolamine
Tolazoline
Others
Ketanserin
Chlorpromazine
ii) α1
Selective
Prazosin
Doxazosin
Terazosin
Tamsulosin
Alfuzosin
iii) α2
Selective
Yohimbine
2) β Blockers
a)Non-selective
i)
Without intrinsic sympathomimetic activity
Propranolol
Sotalol
Timolol
ii)
With intrinsic sympathomimetic activity
Pindol
b) Cardioselective
(β1)
Atenolol
Acebutolol
Metoprolol
Bisoprolol
Celiprolol
Esmolol
Betaxolol
Nebivolol
c)β2
selective
Butoxamine
3) α
and β blockers
Labetalol
Carvedilol
Adrenergic drugs classification
1) Based on Structure
a)
Catecholamines
i)
Natural
Adrenaline
Noradrenaline
Dopamine
ii)
Synthetic
Isoprenaline
Dobutamine
b) Non
Catecholamines
Ephedrine
Amphetamine
Mephentermine
Phenylephrine
2) Based on Mechanism of Action
a)
Directly acting
Adrenaline
Noradrenaline
Isoprenaline
Phenylephrine
Salbutamol
Methoxamine
Xylometazoline
b)
Indirectly acting
Tyramine
c)
Acting by both mechanisms
Ephedrine
Amphetamine
Mephentermine
3) Based on Spectrum of Activity
a)α
agonists
i) α1
selective
Phenylephrine
ii) α2
selective
Clonidine
b) β
Agonists
i)
Non-selective
Isoprenaline
ii) β1
selective
Dobutamine
iii) β2
selective
Terbutaline
Salbutamol
c) α
and β agonists
Adrenaline
Noradrenaline
d)
Dopamine agonists Dopamine (D1 and D2)
Fenoldopam
4) Clinical/ Therapeutic Classification
a)
Pressor agents
Dopamine
Noradrenaline
Methoxamine
Mephentermine
Phenylephrine
Ephedrine
b)
Cardiac stimulants
Adrenaline
Dobutamine
Isoprenaline
c) CNS
stimulants
Amphetamine
Dexamphetamine
Methamphetamine
d)
Bronchodilators
Adrenaline
Isoprenaline
Salbutamol
Salmeterol
Formoterol
Bambuterol
Fenoterol
Terbutaline
Orciprenaline
Isoetherine
e)Nasal
decongestants
Naphazoline
Xylometazoline
Oxymetazoline
Phenylephrine
Pseudoephedrine
Phenylpropanolamine
Propylhexedrine
f) Uterine
relaxants & vasodilators
Ritodrine
Isoxsuprine
Salbutamol
Terbutaline
g)
Anorectics (appetite suppressants)
Fenfluramine
Dexfenfluramine
Sibutramine
Anticholinergic drugs classifiaction
1) Natural Alkaloids
Atropine
Hyoscine
2) Semi-synthetic Derivatives
Homatropine
Atropine methonitrate
Hyoscine butyl bromide
Ipratropium bromide
Tiotropium bromide
3) Synthetic Compounds
a) Mydriatics
Cyclopentolate
Tropicamide
b) Antisecretory antispasmodics
i) Tertiary amines
Dicyclomine
Oxybutynin
Flavoxate
Pirenzepine
Tolterodine
Telenzepine
Trospium
Solifenacin
Darifenacin
Fesoterodine
ii) Quaternary compounds
Propantheline
Glycopyrrolate
Oxyphenonium
Clidinium
Pipenzolate
c) Antiparkinson
Benzhexol
Biperiden
Benztropine
Procyclidine
Ethopropazine
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