Sunday, November 27, 2016

Anti-adrenergic drugs classification


1) α Blockers
a) Non-equilibrium type
Phenoxybenzamine
b) Equilibrium type
i) Non-selective
Ergot alkaloids and derivatives

Ergotamine
Ergotoxine
Dihydroergotamine (DHE)
Dihydroergotoxine

Imidazolines

Phentolamine
Tolazoline

Others

Ketanserin
Chlorpromazine

ii) α1 Selective

Prazosin
Doxazosin
Terazosin
Tamsulosin
Alfuzosin

iii) α2 Selective
Yohimbine


2) β Blockers
a)Non-selective
i) Without intrinsic sympathomimetic activity

Propranolol
Sotalol
Timolol

ii) With intrinsic sympathomimetic activity
Pindol
b) Cardioselective (β1)

Atenolol
Acebutolol
Metoprolol
Bisoprolol
Celiprolol
Esmolol
Betaxolol
Nebivolol

c)β2 selective
Butoxamine

3) α and β blockers

Labetalol
Carvedilol

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