Sunday, November 27, 2016

Cholinergic drugs classification


1) Directly Acting
a) Choline esters


Acetylcholine
Bethanechol
Carbachol
Methacholine


b) Natural Alkaloids


Nicotine
Pilocarpine
Muscarine
Arecoline



2) Indirectly Acting (Cholineesterase inhibitors)
a) Reversible
i) Carbamates


Neostigmine
Physostigmine
Edrophonium 
Pyridostigmine
Ambenonium
Rivastigmine
Galantamine
Donepezil
Rivastigmine


ii) Acridine
Tacrine


b) Irreversible
i) Carbamates
Propoxur
ii) Organophosphates
Echothiophate
Malathion
Dyflos (DFP)
Diazinon
Tabun
Sarin
Soman



3) Cholineesterase reactivators
Pralidoxime
Obidoxime

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